The aza-Diels-Alder reaction of substituted indole 2-carboxaldehydes with Danishefsky's diene has been investigated. The reaction proceeds with a high degree of diastereoselectivity providing highly functionalized 2-(2-piperidyl)indoles which are further elaborated into novel polycyclic heterocycles.
|Original language||English (US)|
|Number of pages||4|
|State||Published - Jan 1 2002|
All Science Journal Classification (ASJC) codes
- Drug Discovery
- Organic Chemistry