An improved protocol for the preparation of 3-pyridyl- and some arylboronic acids

Wenjie Li, Dorian P. Nelson, Mark S. Jensen, R. Scott Hoerrner, Dongwei Cai, Robert D. Larsen, Paul J. Reider

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179 Scopus citations

Abstract

3-Pyridylboronic acid was prepared in high yield and bulk quantity from 3-bromopyridine via a protocol of lithium-halogen exchange and "in situ quench". This technique was further studied and evaluated on other aryl halides in the preparation of arylboronic acids.

Original languageEnglish (US)
Pages (from-to)5394-5397
Number of pages4
JournalJournal of Organic Chemistry
Volume67
Issue number15
DOIs
StatePublished - Jul 26 2002
Externally publishedYes

All Science Journal Classification (ASJC) codes

  • Organic Chemistry

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    Li, W., Nelson, D. P., Jensen, M. S., Hoerrner, R. S., Cai, D., Larsen, R. D., & Reider, P. J. (2002). An improved protocol for the preparation of 3-pyridyl- and some arylboronic acids. Journal of Organic Chemistry, 67(15), 5394-5397. https://doi.org/10.1021/jo025792p