A general procedure for the synthesis of substituted phenylacetylpyridines in excellent yields is described using a Horner-Emmons condensation between α-aminoalkylphosphonates of pyridinecarboxaldehydes and benzaldehydes with cesium carbonate at room temperature.
|Original language||English (US)|
|Number of pages||4|
|State||Published - Mar 26 1998|
All Science Journal Classification (ASJC) codes
- Drug Discovery
- Organic Chemistry