@article{4bf051cc24464483bdf1af565f9e3fbc,
title = "An expedient synthesis of maraviroc (UK-427,857) via C-H functionalization",
abstract = "Abstract A new, concise synthesis of the CCR-5 receptor antagonist maraviroc (UK-427,857) from 3-phenyl-1-propanol has been completed in four steps featuring a site-selective C-H functionalization.",
keywords = "Amination, C-H functionalization, CCR-5, HIV/AIDS, Maraviroc",
author = "Bedell, {T. Aaron} and Hone, {Graham A.B.} and {Du Bois}, Justin and Sorensen, {Erik J.}",
note = "Funding Information: The authors would like to thank Dr. David A. Price and Dr. David Edmonds of Pfizer for helpful discussions and Pfizer for the generous gift of the tosylate salt of compound 6 . This work was supported by the National Institute of General Medical Sciences ( GM065483 ), CCI Center for Selective C–H Functionalization National Science Foundation ( CHE-1205646 ), and Princeton University . Publisher Copyright: {\textcopyright} 2015 Elsevier Ltd.",
year = "2015",
month = may,
day = "25",
doi = "10.1016/j.tetlet.2015.01.074",
language = "English (US)",
volume = "56",
pages = "3620--3623",
journal = "Tetrahedron Letters",
issn = "0040-4039",
publisher = "Elsevier Limited",
number = "23",
}