An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains

K. M.J. Brands; G. Marchesini; J. M. Williams; U. H. Dolling; P. J. Reider

doi:10.1016/0040-4039(96)00447-9

An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains

K. M.J. Brands, G. Marchesini, J. M. Williams, U. H. Dolling, P. J. Reider

Research output: Contribution to journal › Article › peer-review

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Abstract

A convenient and high yielding one-pot process for the preparation of protected 2-thia-5-azabicyclo-[2.2.1]heptan-3-ones from 4-hydroxyproline and their use in the synthesis of carbapenem sidechains is described.

Original language	English (US)
Pages (from-to)	2919-2922
Number of pages	4
Journal	Tetrahedron Letters
Volume	37
Issue number	17
DOIs	https://doi.org/10.1016/0040-4039(96)00447-9
State	Published - Apr 22 1996
Externally published	Yes

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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title = "An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains",

abstract = "A convenient and high yielding one-pot process for the preparation of protected 2-thia-5-azabicyclo-[2.2.1]heptan-3-ones from 4-hydroxyproline and their use in the synthesis of carbapenem sidechains is described.",

author = "Brands, \{K. M.J.\} and G. Marchesini and Williams, \{J. M.\} and Dolling, \{U. H.\} and Reider, \{P. J.\}",

year = "1996",

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language = "English (US)",

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AU - Brands, K. M.J.

AU - Marchesini, G.

AU - Williams, J. M.

AU - Dolling, U. H.

AU - Reider, P. J.

PY - 1996/4/22

Y1 - 1996/4/22

N2 - A convenient and high yielding one-pot process for the preparation of protected 2-thia-5-azabicyclo-[2.2.1]heptan-3-ones from 4-hydroxyproline and their use in the synthesis of carbapenem sidechains is described.

AB - A convenient and high yielding one-pot process for the preparation of protected 2-thia-5-azabicyclo-[2.2.1]heptan-3-ones from 4-hydroxyproline and their use in the synthesis of carbapenem sidechains is described.

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U2 - 10.1016/0040-4039(96)00447-9

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AN - SCOPUS:0030007322

SN - 0040-4039

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SP - 2919

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JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 17

ER -

An expedient one-pot synthesis for protected 2-thia-5-azabicyclo[2.2.1]heptan-3-ones. Versatile intermediates in the synthesis of carbapenem sidechains

Abstract

All Science Journal Classification (ASJC) codes

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